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Classes of Antiretroviral Drugs











































































































TABLE 59-5. Classes of Antiretroviral Drugs
Drug Class
Categorya
Nucleoside reverse transcriptase inhibitors
  Abacavir
C
  Didanosine
B
  Emtricitabine
B
  Lamivudine
C
  Stavudine
C
  Tenofovir
B
  Zalcitabine
C
  Zidovudine
C
Non-nucleoside reverse transcriptase inhibitors
  Delavirdine
C
  Efavirenz
C
  Nevirapine
C
Protease inhibitors
  Amprenavir
C
  Atazanavir
B
  Fosaprenavir
C
  Indinavir
C
  Lopinavir/ritonavir
C
  Nelfinavir
B
  Ritonavir
B
  Saquinavir
B
Fusion inhibitors
  Enfuvirtide
B
aFDA pregnancy category classification—see Chapter 14
(p. 344).
From U.S. Public Health Service (2004a).